Basic Peptide Information

DICL ID
DICL_Pep_06332
Ion Channel
Neuronal acetylcholine receptor subunit alpha-9/alpha-10
Peptide Function
Antagonist
Gene Name
CHRNA9/CHRNA10

Activity Data (nM)

IC50
30 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified

Sequence Information

Peptide Sequence
GCCSHPACSVNHPELC
Peptide UniProt Accession
Not available
UniParc
UPI0001874811
Peptide Synonyms/Alias
[CHEMBL3104239; BDBM50445326]
Peptide Species
Not specified
Peptide Name
Not available
CAS Number
Not available

Experimental Conditions

pH
pH 7.4
Holding Potential (mV)
−70 mV
Temperature
Room Temperature
Test Method
Patch-clamping
Test Species
Not specified

Binding Information

Binding Site
Extracellular domain
Binding Site Residue
Not specified

Ion Channel Information

Gene Abbreviation (ABB)
nAChRs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)

References & Disease Information

Disease
Not specified
PubChem CID
URL
Not available
PMID
Patent
Not available